Aza-Diels-Alder reaction of α,β-unsaturated sulfinylimines derived from α-amino acids with enolethers and enamines
- Egileak:
- Francisco Palacios, Javier Vicario, Domitila Aparicio
- Urtea:
- 2007
- Aldizkaria:
- Tetrahedron Letters
- Liburukia:
- 48
- Hasierako orria - Amaierako orria:
- 6747 - 6750
- Deskribapena:
-
α,β-Unsaturated sulfinylimines derived from α-amino acids undergo aza-Diels–Alder reaction with electron rich dienophiles such as enolethers and enamines. Subsequent elimination of sulfinyl and amine or alkoxy moiety on the resulting cycloadducts affords pyridines derived from α-amino acids.